Avorelin

Avorelin has been in phase II clinical trials by Mediolanum for the treatment of prostate cancer, breast cancer and endometriosis. However, this research has been discontinued.

General Information

Update Date:2016-04-22

Drug Name:
Avorelin
Research Code:
EP-23904; MF-6001
Trade Name:
MOA:
Luteinizing hormone releasing hormone (LH-RH) agonist
Indication:
Prostate cancer; Breast cancer; Endometriosis
Status:
Phase Ⅱ (Discontinued)
Company:
Mediolanum (Originator)
Sales:
ATC Code:
Chemical Structure

Update Date:2016-02-15

Molecular Weight 1296.48
Formula C65H85N17O12
CAS No. 140703-49-7 (Avorelin);
Chemical Name 1-9-Luteinizing hormone-releasing factor (swine), 6-(2-methyl-D-tryptophan)-9-(N-ethyl-L-prolinamide)-
Avorelin (Free Acid/Base)Parameters:
MW HD HA FRB* PSA* cLogP*
1296.48 18 29 34 445 0.926±0.984
*:Calculated by ACD/Labs software V11.02.